[Code of Federal Regulations]
[Title 21, Volume 4]
[Revised as of April 1, 2001]
From the U.S. Government Printing Office via GPO Access
[CITE: 21CFR250.201]

[Page 152-153]
 
                        TITLE 21--FOOD AND DRUGS
 
CHAPTER I--FOOD AND DRUG ADMINISTRATION, DEPARTMENT OF HEALTH AND HUMAN 
                                SERVICES
 
PART 250--SPECIAL REQUIREMENTS FOR SPECIFIC HUMAN DRUGS--Table of Contents
 
               Subpart C--Requirements for Drugs and Foods
 
Sec. 250.201  Preparations for the treatment of pernicious anemia.


    (a) The ninth announcement of the Anti-anemia Preparations Advisory 
Board of the United States Pharmacopeia is concerned with the status of 
the treatment of pernicious anemia. It clearly presents the following 
facts:
    (1) The Sixteenth Revision of the Pharmacopeia of the United States, 
which became official on October 1, 1960, does not include preparations 
intended for the treatment of pernicious anemia by oral administration.
    (2) The U.S.P. unit for anti-anemia preparations no longer has any 
significance.
    (3) The U.S.P. Anti-anemia Preparations Advisory Board was 
disbanded.
    (b) On the basis of the scientific evidence and conclusions 
summarized in the statement of the U.S.P. Anti-anemia Preparations 
Advisory Board as well as pertinent information from other sources, the 
Commissioner of Food and Drugs finds it is the consensus of well 
informed medical opinion that:
    (1) The parenteral administration of cyanocobalamin or vitamin 
B12 is generally recognized as a fully effective treatment of 
pernicious anemia. Parenteral cyanocobalamin preparations have not been 
and are not authorized for use except by or on the prescription of a 
duly licensed medical practitioner.
    (2) Some patients afflicted with pernicious anemia do not respond to 
orally ingested products. There is no known way to predict which 
patients will fail to respond or will cease to respond to the treatment 
of pernicious

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anemia with orally ingested preparations.
    (3) The substitution of a possibly inadequate treatment, such as the 
ingestion of oral preparations of vitamin B12 with intrinsic 
factor concentrate, in place of parenteral vitamin B12 
products for a disease condition as serious as pernicious anemia cannot 
be regarded as safe in all cases.
    (4) The development of the classical symptoms of pernicious anemia 
that would cause a person to seek medical attention may in some cases be 
delayed by oral ingestion of intrinsic factor. Pernicious anemia is a 
disease that is associated, among other things, with a higher than 
normal incidence of cancer of the stomach and that for the safety of the 
patient, requires continuous expert medical supervision.
    (5) With inadequate treatment there may be markedly deleterious 
effects on the nervous system. It is well established that whereas the 
development of anemia is completely reversible with adequate treatment, 
the involvement of the nervous system may not be completely reversible 
and thus may result in permanent damage.
    (6) Some hematologists prescribe oral preparations of vitamin 
B12 in the treatment of pernicious-anemia patients.
    (7) Intrinsic factor and intrinsic factor concentrate serve no known 
useful therapeutic or nutritive purpose except to the extent that they 
do increase the gastrointestinal absorption of vitamin B12 in 
patients with a deficiency or absence of intrinsic factor, which may 
eventually lead to pernicious anemia. This conclusion does not apply to 
diagnostic procedures using radioactive cyanocobalamin.
    (8) Medical expertise is required for the diagnosis as well as the 
management of pernicious anemia.
    (c) The Eleventh Edition of The National Formulary and its first 
Interim Revision include monographs for oral preparations of vitamin 
B12 with intrinsic factor concentrate, establish a unit of 
vitamin B12 with intrinsic factor concentrate, and provide 
for a National Formulary Anti-anemia Preparations Advisory Board to 
assign the potency of such preparations. This provides for the 
availability of such oral preparations, standardized within the meaning 
of the broad limits characteristic of the evaluation of such 
preparations.
    (d) Any drug that is offered for or purports to contain intrinsic 
factor or intrinsic factor concentrate will be regarded as misbranded 
within the meaning of section 503(b) of the Federal Food, Drug, and 
Cosmetic Act unless it is labeled with the legend ``Caution--Federal law 
prohibits dispensing without prescription.''
    (e) Any drug for oral ingestion intended, represented, or advertised 
for the prevention or treatment of pernicious anemia or which purports 
to contain any substance or mixture of substances described in paragraph 
(d) of this section (other than diagnostic drugs containing radioactive 
cyanocobalamin) will be regarded as misbranded under sections 502 (f)(2) 
and (j) of the act unless its labeling bears a statement to the effect 
that some patients afflicted with pernicious anemia may not respond to 
the orally ingested product and that there is no known way to predict 
which patients will respond or which patients may cease to respond to 
the orally ingested products. The labeling shall also bear a statement 
that periodic examinations and laboratory studies of pernicious anemia 
patients are essential and recommended.
    (f) Under section 409 of the Federal Food, Drug, and Cosmetic Act, 
intrinsic factor and intrinsic factor concentrate are regarded as food 
additives. No food additive regulation nor existing extension of the 
effective date of section 409 of the act authorizes these additives in 
foods, including foods for special dietary uses. Any food containing 
added intrinsic factor or intrinsic factor concentrate will be regarded 
as adulterated within the meaning of section 402(a)(2)(C) of the act.
    (g) Regulatory action may be initiated with respect to any article 
shipped within the jurisdiction of the act contrary to the provisions of 
this policy statement after the 180th day following publication of this 
statement in the Federal Register.

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